Wednesday, October 2nd
13:30 Registration
15:30 OpeningCoral Barbas, Vicechancellor of
Research, CEU-USP; Beatriz de Pascual-Teresa,
Organizing Committee, CEU-USP; Antoni Torrens,
President SEQT
ChairpersonJavier Rojo/Antoni Torrens
16:00 Inaugural Lecture: "Antibody-Based
Therapeutics for Cancer Therapy"
Peter Senter, Seattle Genetics, EEUU
17:00 IS1: “Synthetic biology and smart
therapeutic systems”
Guillermo de la Cueva Méndez (BIONAD- Centro Andaluz
de Nanomedicina y Biotecnología, Málaga, Spain)
17:30 IS2: “Glycofullerenes for
Biological Applications”
Nazario Martín León (Universidad Complutense de
Madrid, Spain)
18:00 SEQT Awards
18:30 OC1: “A new strategy to gain
selectivity within the gelatinases subfamily”
Benjamin Fabre. (Universidad CEU San Pablo, Madrid,
Spain) Ramón Madroñero SEQT Award
20:00 Welcome Cocktail
Thursday, October 3rd
MORNING SESSION
Chairperson:
Mª José Camarasa/Mª Luz López
09:00 IS3: “3D Pharmacophore Models:
Efficient Tools for Hit Identification,Lead
Optimization, and Ligand Profiling”
Thierry Langer (Prestwick Chemical, Illkirch, France)
09:30 IS4: “Integrating Intramolecular
Hydrogen Bonding (IMHB) considerations in Drug
Discovery using lipophilicity as a Tool”
Giulia Caron (University of Turin, Italy)
10:00 IS5: “Nucleic acids in
G-quadruplex conformations as innovative targets
against cancer”
Stefano Alcaro (Universitá "Magna Graecia",
Catanzaro, Italy)
10:30 Coffee Break
11:00 IS6: “ORL-1 Antagonists: Lead
Optimization and PET Tracer Development”
Angeles Martínez Grau (Lilly, S.A., Madrid, Spain)
11:30 IS7: “The asymmetric architecture
of G protein-coupled receptor heteromers with G
proteins explains signalling cross-talk”
Peter McCormick (Universidad de Barcelona)
12:00 Oral Communications
Communications (OC2-OC5)
OC2: “Synthesis and Pharmacological
Evaluation of Acetaminophen Analogues with
Antinociceptive Properties”
Pilar Goya (Instituto de Química Médica, CSIC, Madrid,
Spain)
OC3: “Synthesis and Pharmacological
Evaluation of Acetaminophen Analogues with
Antinociceptive Properties”
Pilar Goya (Instituto de Química Médica, CSIC, Madrid,
Spain)
OC3:“Applications of click chemistry in
sphingolipid research”
Antonio Delgado (IQAC-CSIC, Barcelona, Spain)
OC4:“Computational chemistry for
identifying differences among choline kinases active
sites”
Lucía Serrán Aguilera (Universidad de Granada, Spain)
OC5:“Impact of fluorination on
proteolytic stability of peptides: a case study using
α-chymotrypsin and pepsin”
Jeremie Mortier (Free University of Berlin, Germany)
13:00 Lunch
AFTERNOON SESSION
Chairperson: Pilar Goya/Julio Álvarez Builla
15:00 IS8: : “Amino Acid-Derived
β–Lactams: Synthesis, Biological Activity and
Beyond”
Rosario González Muñiz (Instituto de Química Médica,
CSIC, Madrid, Spain)
15:30 OC6: “New non-metathetic processes
catalysed by ruthenium complexes for the synthesis of
heterocycles”
Javier Pérez-Castells (Universidad CEU San Pablo,
Madrid, Spain)
15:45:Poster Session and Coffee
16:45 Oral Communications (OC7-OC8)
OC7: “Merging of pineal neurochemicals.
pharmacological profiles and neurogenic
potential”
Mario de la Fuente Revenga (Instituto de Química
Médica, CSIC, Madrid, Spain)
OC8:“Drugging the von hippel lindau E3
ubiquitin ligase: potential drugs and useful chemical
tools”
Carles Galdeano (University of Dundee, Dundee, UK)
19:30 Cultural evening:
"Discover most unknown Madrid`s old town,even for
locals; in a 1,30-1,45 hrs aprox walking tour seeing
highlights bringing back its ancient
past,legends,alleyways,monuments and curiosities with
a fully licensed guides that will make you travel
through the time" Underground: Puerta del Sol
metro station.
Friday, October 4th
MORNING SESSION
ChairpersonJordi Gracia/Javier Fernández Gadea
09:00 IS9: “Next-Generation Inhibitors
for Kinases, Histone-Deacetylases, and Histone
Methyltransferases: The discovery of
Slowness”
Gerhard Müller (Mercachem, The Netherlands)
09:30 IS10:“Exploring the kinome with
kinase broad screening”
Gary Tresadern (Janssen R&D, Beerse, Belgium)
10:00 IS11“Antibiotic Treatment of
Tuberculosis: Old Problems, New Solutions”
Mónica Cacho Izquierdo (GlaxoSmithKline, Madrid,
Spain)
10:30 Coffee Break
11:00 Oral Communications (OC9-OC12)
OC9: "Design of mycobacterium tuberculosis
shikimate kinase inhibitors inspired by the enzymatic
movements for catalytic turnover”
Verónica Prado (CIQUS, Universidad de Santiago de
Compostela, Spain)
OC10: “From hit to lead in search of new
inhibitors of the enzyme isoprenylcysteine carboxyl
methyltransferase (ICMT)”
Silvia Ortega-Gutiérrez (Universidad Complutense,
Madrid, Spain)
OC11:“Design, synthesis and biological
evaluation of cyclic acylguanidines as bace-1
inhibitors: effect of ring size on activity and
selectivity versus BACE-2”
Myriam Ciordia (Janssen Pharmaceutical Research &
Development, Toledo, Spain)
OC12: “-Omics tools for studying changes
in metabolic pathways of new drugs”
Isidre Masana (Agilent Technologies)
12:00 SEQT Meeting
13:00 Lunch
AFTERNOON SESSION
ChairpersonConcepción González Bello/Antonio
Pineda
15:00 IS12:“ETP-CNIO Academic Early Drug
Discovery: PIM Kinase Inhibitors”
Joaquín Pastor (CNIO- Centro Nacional de
Investigaciones Oncológicas, Madrid, Spain)
15:30 OC13“Different levels of apoptosis
caused by enantiomers in breast cancer cells”
Joaquín M. Campos (Universidad de Granada, Spain)
15:45: Poster Session and Coffee
16:45 Oral Communications (OC14-OC16)
OC14:“Tumor vascular disrupting agents:
identification and optimization of novel
hits”
Mª Dolores Canela (Instituto de Química Médica,
CSIC, Madrid, Spain)
OC15:“3-Substituted indole derivatives as
antimitotic agents”
Raquel Álvarez Lozano (Universidad de Salamanca,
Salamanca, Spain)
OC16:“Chemical biology for drug
discovery: two case studies in drug
repurposing”
Jordi Quintana (Parc Científic de Barcelona, Spain)
17:30 Concluding Remarks. Poster and Oral
Communication Awards
21:00 Gala Dinner
Gala dinner will be held in "La Posada de la
Villa”, a classic Spanish restaurant in Madrid.
It is included in the distinguished Michelin Guide)
and has been awarded in many occasions: Grand Collar
Gourmet, the Chaîne des Rotisseurs, etc.
Posada de la Villa Restaurant C/ Cava Baja, 9.
Underground: La Latina metro station.
Important information about posters:
-
Poster session 1: Thursday October 3rd
15:45-16:45: ODD numbers
-
Poster session 1: Friday October 4th
15:45-16:45: EVEN numbers